Custom-tailored

end-to-end services.

We offer syntheses of KSMs, RSMs, advanced intermediates in compliance with the latest regulatory requirements with affordable costs and high quality.

Contract Manufacturing of Intermediates and Drug Substances

Technical and regulatory support

A dedicated team of technical and regulatory experts to support you.

Added Value

Complimentary services such as intellectual property, quality management, regulatory affairs, logistics (import, export), etc.

Scale-up

No limitations of chemistry, technology, or volumes

INTERMEDIATESList

API Name CAS Number Intermediate Name Status
Linagliptin 666816-98-4 8-Bromo-7-(2-butynyl)-3,7-dihydro-3-methyl-1H-purine-2,6-dione Commercialised
Linagliptin 109113-72-6 2-(Chloromethyl)-4-methylquinazoline Commercialised
Linagliptin 309956-78-3 (R)-3-(Boc-Amino) piperidine Under Development
Rivaroxaban 161596-47-0 (S)-2-(oxiran-2-ylmethyl isoindoline-1,3-dione (or) (S)-Glycidylphthalimide Commercialised
Rivaroxaban 438056-69-0 4-(4-Aminophenyl) morpholin-3-one Commercialised
Rivaroxaban 24065-33-6 5-Chlorothiophene-2-Carboxylic acid Commercialised
Vildagliptin 207557-35-5 (2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile Commercialised
Vildagliptin 702-82-9 3-Amino-1-adamantanol Commercialised
Bilastine 17178-11-9 2-Ethoxyethyl 4-methyl benzenesulfonate Commercialised
Bilastine 38385-95-4 2-Piperdin-4-yl-1H-Benzimidazole Commercialised
Bilastine 953071-73-3 Tert-butyl 4-(1H-benzo[d]imidazol-2-yl) piperidine-1-carboxylate Commercialised
Bilastine 1841081-72-8 1-(2-Ethoxyethyl)-2-(piperidin-4-yl)-1H-benzo[d]imidazole hydrochloride Commercialised
Bilastine 202189-77-3 2-(2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d] imidazol-2-yl) piperidin-1-yl) ethyl) phenyl) propan-2-yl)-4,4-dimethyl-4,5-dihydrooxazole Commercialised
Mirabegron 66659-20-9 2-Amino-4-thiazoleacetic acid hydrochloride Tech pack available
Ticagrelor 145783-15-9 4,6-Dichloro-2-(propylthio)-5-pyrimidinamine Tech pack available
Niraparib 1476776-55-2 tert-Butyl (S)-3-(4-bromophenyl)
piperidine-1-carboxylate
Tech pack available

INTERMEDIATESUNDER DEVELOPMENT

API Name CAS Number Intermediate Name Status
Apixaban   5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone Feasibility completed
Apixaban   Chloro[(4-methoxyphenyl) hydrazono]- acetic acid ethyl ester Feasibility completed
Empagliflozin   (S)-(5-Bromo-2-chlorophenyl) (4-((tetrahydrofuran-3-yl)oxy)phenyl)methanone Under tech transfer
Empagliflozin   (S)-3-(4-(5-Bromo-2-chlorobenzyl) phenoxy) tetrahydrofuran Under tech transfer
Dapagliflozin   (5-Bromo-2-chlorophenyl) (4-ethoxyphenyl) methanone Optimisation in progress
Dapagliflozin   5-Bromo-2-chloro-4’-ethoxydiphenylmethane Optimisation in progress
Sitagliptin   (R)-N-Boc-3-Amino-4-(2,4,5-trifluorophenyl) butanoic acid Feasibility in progress
Sitagliptin   3-(Trifluoromethyl)-5,6,7,8-tetrahydro [1,2,4] triazolo[4,3-a] pyrazine. HCl Feasibility in progress
Sitagliptin Methyl 4-(2,4,5-trifluorophenyl)-3-oxobutanoate Optimisation completed
Oseltamivir   Ethyl (1S,5R,6S)-5-(1-ethylpropoxy)-7-oxabicyclo [4.1.0] hept-3-ene-3-carboxylate Optimisation completed
Amlodipine   Phthaloyl amlodipine Optimisation completed
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